Volume One
HETEROCYCLIC COMPOUNDS: AN INTRODUCTION
Heterocyclic Compounds: An Introduction
Structure and Reactivity of Aromatic Five-Membered Systems
Structure and Reactivity of Aromatic Six-Membered Systems
Basic Literature on Heterocyclic Compounds
THREE-MEMBERED HETEROCYCLES: STRUCTURE AND REACTIVITY
Aziridines
2H-Azirines
Oxiranes
Thiiranes
Diaziridines
3H-Diazirines
Oxaziridines
Dioxiranes
FOUR-MEMBERED HETEROCYCLES: STRUCTURE AND REACTIVITY
Azetidines
Oxetanes
Thietanes
Other Four-Membered Heterocycles
FIVE-MEMBERED HETEROCYCLES: PYRROLE AND RELATED SYSTEMS
Introduction
General Reactivity
Relevant Natural and/or Useful Compounds
Pyrrole Ring Synthesis
Reactivity
Pyrrole Derivatives
Addendum
FIVE-MEMBERED HETEROCYCLES: INDOLE AND RELATED SYSTEMS
Introduction
General Properties
Relevant Natural and/or Useful Compounds
Indole Synthesis
Reactivity of Indole
Chemistry of Indole Derivatives
Addendum
FIVE-MEMBERED HETEROCYCLES: FURAN
Introduction
Synthesis of Furans
Reactivity
Oxyfurans and Aminofurans
Addendum
FIVE-MEMBERED HETEROCYCLES: BENZOFURAN AND RELATED SYSTEMS
Introduction
General Structure and Reactivity
Isolation of Naturally Occurring Benzofurans
Synthesis of Benzofuran
Uses of Benzofuran
Volume Two
FIVE-MEMBERED HETEROCYCLES: 1,2-AZOLES. PART 1. PYRAZOLES
Introduction
General Reactivity
Relevant Natural and/or Useful Compounds
Synthesis of Pyrazoles and Indazoles
Reactivity
Derivatives
FIVE-MEMBERED HETEROCYCLES: 1,2-AZOLES. PART 2. ISOXAZOLES
Introduction
General Reactivity
Relevant Natural and/or Useful Compounds
Synthesis of Isoxazoles and Isothiazoles
Synthesis of Benzisoxazoles and Benzisothiazoles
Reactivity of 1,2-Azoles
FIVE-MEMBERED HETEROCYCLES: 1,2-AZOLES
Introduction
General Reactivity
Synthesis of Aromatic 1,3-Azoles
Reactivity
Derivatives
FIVE-MEMBERED HETEROCYCLES WITH TWO HETEROATOMS: O AND S DERIVATIVES
Introduction
1,2-Dioxoles and 1,2-Dioxolanes
1,3-Dioxoles and 1,3-Dioxolanes
1,2-Dithioles and 1,2-Dithiolanes
1,3-Dithioles and 1,3-Dithiolanes
1,2-Oxathioles and 1,2-Oxathiolanes
1,3-Oxathioles and 1,3-Oxathiolanes
FIVE-MEMBERED HETEROCYCLES WITH THREE HETEROATOMS: TRIAZOLES
1,2,3-Triazoles
Benzotriazole
1,2,4-Triazoles
OXADIAZOLES
Introduction
1,2,3-Oxadiazoles
1,2,4-Oxadiazoles
1,2,5-Oxadiazoles
1,3,4-Oxadiazoles
Volume Three
THIADIAZOLES
Introduction
1,2,3-Thiadiazoles
1,2,4-Thiadiazoles
1,3,4-Thiadiazoles
FIVE-MEMBERED HETEROCYLCES WITH FOUR HETEROATOMS: TETRAZOLES
Introduction
Synthetic Methods
Reactions of Tetrazoles
SIX-MEMBERED HETEROCYCLES: PYRIDINES
Introduction
Synthesis of Pyridines
Reactivity
Pyridine Derivatives
Appendix
SIX-MEMBERED HETEROCYCLES: QUINOLINE AND ISOQUINOLINE
Quinoline
Isoquinoline
SIX-MEMBERED RINGS WITH ONE OXYGEN: PYRYLIUM ION, RELATED SYSTEMS AND BENZO-DERIVATIVES
Introduction
Pyrylium Cation and Benzo-Derivatives
2H-Pyrans and 4H-Pyrans
Pyrones, Coumarins, and Chromones
SIX-MEMBERED HETEROCYCLES: 1,2-, 1,3-, AND 1,4-DIAZINES
Introduction
General Reactivity
Relevant Natural/Biological Compounds
Synthesis of Pyridazines (1,2-Diazines)
Synthesis of Pyrimidines (1,3-Diazines)
Synthesis of Pyrazines (1,4-Diazines)
Reactivity of Diazines
Important Derivatives
SIX-MEMBERED HETEROCYCLES: TRIAZINES, TETRAZINES AND OTHER POLYAZA SYSTEMS
Introduction
1,2,3-Triazines
1,2,4-Triazines
1,3,5-Triazines
Tetrazines
Volume Four
SEVEN-MEMBERED HETEROCYCLES: AZEPINES, BENZO DERIVATIVES AND RELATED SYSTEMS
Introduction
Relevant Natural and Useful Compounds
Relevated Computational Chemistry, Physicochemical, and Spectroscopic Data
Valence Tautomerism in Seven-Membered Heterocycles
Synthesis
Reactivity of Azepines
Reactivity of Oxepines
Reactivity of Thiepines
HETEROCYCLES CONTAINING A RING-JUNCTION NITROGEN
Introduction
Pyrrolizines
Indolizines
Quinolizinium Salts
PHOSPHORUS HETEROCYCLES
Introduction
Phospholes
Phosphinines
Other P Heterocycles
Applications of Phosphorus Heterocycles
Addendum
THE CHEMISTRY OF 2-AZETIDINONES (BETA-LACTAMS)
Monocyclic Derivatives
Penicillins and Cephalosporins
THE CHEMISTRY OF BENZODIAZEPINES
Introduction
Relevant Benzodiazepines
1,4-Benzodiazepines: General Synthetic Methods
Modifications of the 1,4-Benzodiazepine Ring
1,4-Benzodiazepines with a Fused Heterocycle
Pyrrolo[2,1-c][1,4]Benzodiazepines (PBDs)
1,5-Benzodiazepines
2,3-Benzodiazepines
PORPHYRINS: SYNTHESES AND REACTIONS
Introduction
Synthetic Chemistry of Porphyrins and Expanded Porphyrins
Reactivity of Porphyrins
NEW MATERIALS DERIVED FROM HETEROCYCLIC SYSTEMS
Introduction
Color and Fluorescent Agents
Self-Assembling Materials and Molecular Containers
Unnatural Enzyme Models
Organic Conductors
SOLID PHASE AND COMBINATORIAL CHEMISTRY IN THE HETEROCYCLIC FIELD
Introduction
Solid Supports
Linkers for Solid-Phase Organic Synthesis
Heterocyclic Synthesis on Solid-Phase
